tacrolimus ophthalmic

Off-label use

Description

Tacrolimus ophthalmic suspension is a calcineurin inhibitor used off-label for severe allergic eye diseases including vernal conjunctivitis. It provides potent anti-inflammatory effects by inhibiting T-cell activation and cytokine production. Studies have shown efficacy in steroid-resistant cases of vernal keratoconjunctivitis.

Indications & Therapeutic Use

vernal keratoconjunctivitis, atopic keratoconjunctivitis, severe allergic conjunctivitis

Linked Diseases:

Global Availability (5 countries)

CountryAccess RouteRegulatory PathwayLead TimeStatus

Available Through

This drug is available for procurement through the following fulfilment partner.

Fulfilment Partner
tacrolimus ophthalmic
Generic Nametacrolimus ophthalmic
Active Ingredienttacrolimus
Drug Classvernal keratoconjunctivitis
Manufacturervarious
Dosage Formsophthalmic suspension 0.03%, 0.1%
Medical CodeS01XA20
Orphan StatusNo
Cold ChainNot Required
Lead Time10 days
Reg. StatusOff-label use
Clinical TrialNCT01751126
Countries5 countries
Authority Signals
Last Verified3/21/2026
Data ConfidenceHigh (AI + Pharmacist)
Source Citations6 Validated Nodes