imatinib mesylate

Orphan DrugFDA Approved, EMA Approved

Description

Imatinib is a tyrosine kinase inhibitor that targets BCR-ABL, c-KIT, and PDGFR. It is used in the treatment of various hematologic malignancies and has shown efficacy in systemic mastocytosis including urticaria pigmentosa. The drug works by blocking abnormal protein signaling in affected cells.

Indications & Therapeutic Use

chronic myeloid leukemia, acute lymphoblastic leukemia, systemic mastocytosis, urticaria pigmentosa, gastrointestinal stromal tumors

Global Availability (9 countries)

CountryAccess RouteRegulatory PathwayLead TimeStatus

Available Through

This drug is available for procurement through the following fulfilment partner.

Fulfilment Partner
imatinib mesylate
Generic Nameimatinib mesylate
Brands1 brand available
Active Ingredientimatinib mesylate
Drug Classchronic myeloid leukemia
ManufacturerNovartis
Dosage FormsOral tablet, 100mg, 400mg
Medical CodeL01EA01
Orphan StatusYes — Orphan Drug
Cold ChainNot Required
Lead Time7 days
Reg. StatusFDA Approved, EMA Approved
Clinical TrialNCT00001459
Countries9 countries
Authority Signals
Last Verified3/21/2026
Data ConfidenceHigh (AI + Pharmacist)
Source Citations10 Validated Nodes