Nitisinone

Orphan DrugFDA Approved

Description

Nitisinone is an orphan drug that inhibits 4-hydroxyphenylpyruvate dioxygenase (HPPD). Originally approved for hereditary tyrosinemia type 1, it has been investigated for oculocutaneous albinism due to its effects on tyrosine metabolism. The drug increases tyrosine levels which may enhance melanin production in certain forms of albinism.

Indications & Therapeutic Use

Hereditary tyrosinemia type 1, investigational use in oculocutaneous albinism

Global Availability (7 countries)

CountryAccess RouteRegulatory PathwayLead TimeStatus

Available Through

This drug is available for procurement through the following fulfilment partner.

Fulfilment Partner
Nitisinone
Generic NameNitisinone
Brands1 brand available
Active IngredientNitisinone
Drug ClassHereditary tyrosinemia type 1
ManufacturerSobi (Swedish Orphan Biovitrum)
Dosage FormsOral capsule, 2mg, 5mg, 10mg, 20mg; Oral suspension, 4mg/mL
Medical CodeA16AX04
Orphan StatusYes — Orphan Drug
Cold ChainNot Required
Lead Time21 days
Reg. StatusFDA Approved
Countries7 countries
Authority Signals
Last Verified3/21/2026
Data ConfidenceHigh (AI + Pharmacist)
Source Citations8 Validated Nodes