Tolvaptan

Orphan DrugFDA Approved

Description

Tolvaptan is a selective vasopressin V2-receptor antagonist indicated for slowing kidney function decline in adults at risk of rapidly progressing autosomal dominant polycystic kidney disease (ADPKD). It has been studied for use in juvenile nephronophthisis due to similar cystic kidney pathology. The drug works by blocking vasopressin receptors in the kidney collecting duct, reducing cyst growth and preserving renal function.

Indications & Therapeutic Use

Autosomal dominant polycystic kidney disease, juvenile nephronophthisis (investigational)

Global Availability (9 countries)

CountryAccess RouteRegulatory PathwayLead TimeStatus

Available Through

This drug is available for procurement through the following fulfilment partner.

Fulfilment Partner
Tolvaptan
Generic NameTolvaptan
Brands1 brand available
Active IngredientTolvaptan
Drug ClassAutosomal dominant polycystic kidney disease
ManufacturerOtsuka Pharmaceutical
Dosage FormsOral tablet 15mg, 30mg, 45mg, 60mg, 90mg
Medical CodeC03XA01
Orphan StatusYes — Orphan Drug
Cold ChainNot Required
Lead Time14 days
Reg. StatusFDA Approved
Clinical TrialNCT01214421
Countries9 countries
Authority Signals
Last Verified3/21/2026
Data ConfidenceHigh (AI + Pharmacist)
Source Citations10 Validated Nodes